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Search Results for " phospholipase a2 "

20

Compounds

Cat No. Product Name Synonyms Targets
T76182 Phospholipase A2
Phospholipase A2 (PLA2), a heat-stable, calcium-dependent enzyme class member, catalyzes the hydrolysis at the sn-2 position of membrane glycerophospholipids, releasing arachidonic acid (AA). It is frequently utilized in...
T17218 Varespladib methyl A-002,LY333013 Others , Phospholipase
Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.
T16751 Rilapladib SB 659032 Phospholipase
Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activating factor receptor.
TN1419 Rhamnetin beta-Rhamnocitrin Others , Phospholipase
Rhamnetin (beta-Rhamnocitrin), a quercetin derivative found in Coriandrum sativum, has antioxidant and anti-inflammatory activities. Rhamnetin inhibits secretory phospholipase A2.
T21907 PACOCF3 1,1,1-trifluoroheptadecan-2-one,Palmityltrifluoromet​hylketone Phospholipase
PACOCF3 (Palmityltrifluoromethylketone) (Palmityltrifluoromet hylketone) is an inhibitor of Ca(2+)-independent phospholipase A2(PLA2) with an IC 50 of 3.8 μM. PACOCF3 alters Ca 2+ signaling in renal tubular cells [1] [2]...
T6109 Darapladib SB-480848 Phospholipase
Darapladib (SB-480848)(IC50=0.25 nM) is a substituted pyrimidone with inhibitory activity towards lipoprotein-associated phospholipase-A2 (Lp-PLA2).
T31204 Darapladib-impurity Others
Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2).
T21815 ONO-RS-082 Others
ONO-RS-082 is a Ca2+-independent phospholipase A2 inhibitor.
T9753 LEI110 Phospholipase
LEI110 is a potent Phospholipase A2, group XVI (PLA2G16) inhibitor with an Ki value of 20 nM. LEI110 is a selective pan-inhibitor of the HRASLS family of thiol hydrolases (i.e., PLA2G16, HRASLS2, RARRES3 and iNAT).
T11874 Lp-PLA2-IN-3 Phospholipase
Lp-PLA2-IN-3 is a potent and orally bioactive lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor that inhibits recombinant human Lp-PLA2 with an IC50 value of 14 nM.
T5454 N-(p-amylcinnamoyl) Anthranilic Acid ACA Phospholipase , TRP/TRPV Channel
N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.
T19729 Dodecylphosphocholine DPC,n C12PC,Foscholine-12,DDPPC,nC12PC,n-C12PC Others
Dodecylphosphocholine (DPC) is a substrate-type inhibitor of pancreas phospholipase A2. Dodecylphosphocholine is a detergent.
T24449 Mepacrine Haffkinine,Erion Others
Mepacrine (Erion) is an acridine derivative formerly widely used as an antimalarial. It is used in cell biological experiments as an inhibitor of phospholipase A2.
T2044 Varespladib LY315920 Phospholipase
Varespladib (LY315920), a specific and effective human non-pancreatic secretory phospholipase A2 (hnsPLA) inhibitor(IC50=7 nM), has been investigated for the treatment and prevention of sickle cell disease, vaso-occlusiv...
T21606L Anti-Inflammatory Peptide 1 Acetate Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base) Phospholipase
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) possesses a potent anti-inflammatory activity in vivo and is a strong inhibitor of phospholipase A2 (PLA2), whose increased presence and activity results in inflammati...
T14689 BMS493 BMS-493 Phospholipase , Retinoid Receptor
BMS493 is an inverse agonist of the pan-retinoic acid receptor (RAR) that inhibits retinoic acid-induced differentiation, enhances the interaction of nuclear co-inhibitors with RARs, attenuates RA signaling, potentiates ...
TN1064 Aristolochic acid C Others
Aristolochic acid C could as the larval feeding stimulants.
TN6993 Benzylideneacetone Benzalacetone Phospholipase , Endogenous Metabolite
Benzylideneacetone, a monoterpene produced by the insect pathogenic bacterium Xenorhabdus nematophila, is a phospholipase A2 (PLA2) inhibitor with inhibitory effects on arachidonoid biosynthesis and enhances baculovirus ...
T0370 Pheniramine maleate Daneral,Inhiston,Trimetose 5-HT Receptor , Histamine Receptor
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of the endothelium-derived re...
T10017 1-Linoleoyl Glycerol Glycerol 1-monolinolate,Monolinolein,Glyceryl monolinoleate,1-Linoleoyl-rac-glycerol Phospholipase
1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots. The (R)-1-Linoleoyl Glycerol and (S)-1-Linoleoyl Glycerol exhibit Lipoprotein-associated phospholipase A2 (...

Compounds

Phospholipase A2
T76182
Synonym:
Target:
Varespladib methyl
T17218
Synonym: A-002,LY333013
Target: Others, Phospholipase
Rilapladib
T16751
Synonym: SB 659032
Target: Phospholipase
Rhamnetin
TN1419
Synonym: beta-Rhamnocitrin
Target: Others, Phospholipase
PACOCF3
T21907
Synonym: 1,1,1-trifluoroheptadecan-2-one,Palmityltrifluoromet​hylketone
Target: Phospholipase
Darapladib
T6109
Synonym: SB-480848
Target: Phospholipase
Darapladib-impurity
T31204
Synonym:
Target: Others
ONO-RS-082
T21815
Synonym:
Target: Others
LEI110
T9753
Synonym:
Target: Phospholipase
Lp-PLA2-IN-3
T11874
Synonym:
Target: Phospholipase
N-(p-amylcinnamoyl) Anthranilic Acid
T5454
Synonym: ACA
Target: Phospholipase, TRP/TRPV Channel
Dodecylphosphocholine
T19729
Synonym: DPC,n C12PC,Foscholine-12,DDPPC,nC12PC,n-C12PC
Target: Others
Mepacrine
T24449
Synonym: Haffkinine,Erion
Target: Others
Varespladib
T2044
Synonym: LY315920
Target: Phospholipase
Anti-Inflammatory Peptide 1 Acetate
T21606L
Synonym: Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base)
Target: Phospholipase
BMS493
T14689
Synonym: BMS-493
Target: Phospholipase, Retinoid Receptor
Aristolochic acid C
TN1064
Synonym:
Target: Others
Benzylideneacetone
TN6993
Synonym: Benzalacetone
Target: Phospholipase, Endogenous Metabolite
Pheniramine maleate
T0370
Synonym: Daneral,Inhiston,Trimetose
Target: 5-HT Receptor, Histamine Receptor
1-Linoleoyl Glycerol
T10017
Synonym: Glycerol 1-monolinolate,Monolinolein,Glyceryl monolinoleate,1-Linoleoyl-rac-glycerol
Target: Phospholipase
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TargetMol